Molecule Details
InChIKeyLCIMOJQEZXDWTA-UHFFFAOYSA-N
Compound Name2-[4-[(4-Anilino-5-nitropyrimidin-2-yl)amino]phenoxy]acetic acid
Canonical SMILESO=C(O)COc1ccc(Nc2ncc([N+](=O)[O-])c(Nc3ccccc3)n2)cc1
Clinical Status Data-mined Candidate
Targets (Human+Pathogen)3
Pfam Stratification Homologous
Avg pChEMBL7.08
SourceChEMBL;BindingDB
2D Structure
2D structure
Activity Profile
Target Activities (3)
Target Gene Organism Category Pfam pChEMBL Type Source
P49840 GSK3A Homo sapiens Human PF00069 7.1 IC50 ChEMBL;BindingDB
O14965 AURKA Homo sapiens Human PF00069 7.1 IC50 ChEMBL;BindingDB
P49841 GSK3B Homo sapiens Human PF00069 7.0 IC50 ChEMBL;BindingDB