Molecule Details
InChIKeyLCBAQTCTQXHTJG-SSDOTTSWSA-N
Compound Name(7R)-2-(2-aminopyrimidin-4-yl)-7-(2-fluoroethyl)-1H,4H,5H,6H,7H-pyrrolo[3,2-c]pyridin-4-one
Canonical SMILESNc1nccc(-c2cc3c([nH]2)[C@H](CCF)CNC3=O)n1
Clinical Status Data-mined Candidate
Targets (Human+Pathogen)3
Pfam Stratification Cross-Family
Avg pChEMBL7.45
SourceBindingDB;ChEMBL
2D Structure
2D structure
Activity Profile
Target Activities (3)
Target Gene Organism Category Pfam pChEMBL Type Source
O00311 CDC7 Homo sapiens Human PF00069 8.3 IC50 ChEMBL;BindingDB
O60563 CCNT1 Homo sapiens Human PF00134 PF21797 7.0 IC50 BindingDB
P50750 CDK9 Homo sapiens Human PF00069 7.0 IC50 ChEMBL