Molecule Details
InChIKeyLASNBXWNXQRYSO-UHFFFAOYSA-N
Compound Name5-hydroxy-1-tosyl-1H-pyrrol-2(5H)-one
Canonical SMILESCc1ccc(S(=O)(=O)N2C(=O)C=CC2O)cc1
Clinical Status Clinical Multi-Target
Targets (Human+Pathogen)3
Pfam Stratification Cross-Family
Avg pChEMBL6.39
SourceBindingDB;ChEMBL;TTD_MultiTarget
2D Structure
2D structure
Activity Profile
Target Activities (3)
Target Gene Organism Category Pfam pChEMBL Type Source
P18505 GABRB1 Homo sapiens Human PF02931 PF02932 6.7 pIC50 TTD_MultiTarget
P00915 CA1 Homo sapiens Human PF00194 6.3 Ki ChEMBL;BindingDB
P00918 CA2 Homo sapiens Human PF00194 6.2 Ki BindingDB