Molecule Details
InChIKeyKZXNHUNTABHMLN-DXPJPUQTSA-N
Compound Namemethyl (10R,14S)-5-amino-14-[4-(3-chloro-2,6-difluorophenyl)-6-oxo-2,3-dihydropyridin-1-yl]-10-methyl-9-oxo-8,16-diazatricyclo[13.3.1.02,7]nonadeca-1(19),2,4,6,15,17-hexaene-4-carboxylate
Canonical SMILESCOC(=O)c1cc2c(cc1N)NC(=O)[C@H](C)CCC[C@H](N1CCC(c3c(F)ccc(Cl)c3F)=CC1=O)c1cc-2ccn1
Clinical Status Data-mined Candidate
Targets (Human+Pathogen)3
Pfam Stratification Homologous
Avg pChEMBL8.33
SourceChEMBL;BindingDB
2D Structure
2D structure
Activity Profile
Target Activities (3)
Target Gene Organism Category Pfam pChEMBL Type Source
P00740 F9 Homo sapiens Human PF00008 PF14670 PF00594 PF00089 8.3 Ki ChEMBL;BindingDB
P03951 F11 Homo sapiens Human PF00024 PF00089 8.3 Ki ChEMBL;BindingDB
P03952 KLKB1 Homo sapiens Human PF00024 PF00089 8.3 Ki ChEMBL;BindingDB