Molecule Details
InChIKeyKZMSAVPDHMHSQO-NRFANRHFSA-N
Compound Name(S)-2-({5-[(1H-Imidazol-4-ylmethyl)-amino]-biphenyl-2-carbonyl}-amino)-4-methyl-pentanoic acid
Canonical SMILESCC(C)C[C@H](NC(=O)c1ccc(NCc2c[nH]cn2)cc1-c1ccccc1)C(=O)O
Clinical Status Clinical Multi-Target
Targets (Human+Pathogen)2
Pfam Stratification Cross-Family
Avg pChEMBL7.05
SourceChEMBL;TTD_MultiTarget
2D Structure
2D structure
Activity Profile
Target Activities (2)
Target Gene Organism Category Pfam pChEMBL Type Source
P49354 FNTA Homo sapiens Human PF01239 7.0 pIC50 TTD_MultiTarget
P53609 PGGT1B Homo sapiens Human PF00432 7.0 IC50 ChEMBL