Molecule Details
InChIKeyKYMADELXCHTVCR-IBGZPJMESA-N
Compound Name(S)-benzyl 1-(2-phenylthiazol-4-yl)-5-(sulfamoylamino)pentylcarbamate
Canonical SMILESNS(=O)(=O)NCCCC[C@H](NC(=O)OCc1ccccc1)c1csc(-c2ccccc2)n1
Clinical Status Clinical Multi-Target
Targets (Human+Pathogen)3
Pfam Stratification Cross-Family
Avg pChEMBL6.2
SourceChEMBL;BindingDB;TTD_MultiTarget
2D Structure
2D structure
Activity Profile
Target Activities (3)
Target Gene Organism Category Pfam pChEMBL Type Source
Q9UBN7 HDAC6 Homo sapiens Human PF00850 PF02148 6.4 IC50 ChEMBL;BindingDB
Q02161 RHD Homo sapiens Human PF00909 6.1 pIC50 TTD_MultiTarget
Q13547 HDAC1 Homo sapiens Human PF00850 6.1 pIC50 TTD_MultiTarget