Molecule Details
InChIKeyKYCYXWHIIAISQF-UHFFFAOYSA-N
Compound Name2-((3-(Difluoromethoxy)pyridin-2-yl)methyl)-7-(4-fluorophenyl)-8-(imidazo[l,2-a]pyridin-6-yl)-[1,2,4 triazolo[l,5-c]pyrimidin-5-amine
Canonical SMILESNc1nc(-c2ccc(F)cc2)c(-c2ccc3nncn3c2)c2nc(Cc3ncccc3OC(F)F)nn12
Clinical Status Data-mined Candidate
Targets (Human+Pathogen)3
Pfam Stratification Homologous
Avg pChEMBL8.76
SourceChEMBL;BindingDB
2D Structure
2D structure
Activity Profile
Target Activities (3)
Target Gene Organism Category Pfam pChEMBL Type Source
P29274 ADORA2A Homo sapiens Human PF00001 10.0 IC50 ChEMBL;BindingDB
P29275 ADORA2B Homo sapiens Human PF00001 8.3 IC50 ChEMBL;BindingDB
P30542 ADORA1 Homo sapiens Human PF00001 8.0 IC50 ChEMBL;BindingDB