Molecule Details
InChIKeyKXZUNTUEDNVFLH-UHFFFAOYSA-N
Compound Name4-[4-[1-(3-Methoxypyrazin-2-yl)-8-[(3-methyl-2-pyridinyl)methyl]-2,4-dioxo-1,3,8-triazaspiro[4.5]decan-3-yl]phenyl]-3-methylbenzoic acid
Canonical SMILESCOc1nccnc1N1C(=O)N(c2ccc(-c3ccc(C(=O)O)cc3C)cc2)C(=O)C12CCN(Cc1ncccc1C)CC2
Clinical Status Data-mined Candidate
Targets (Human+Pathogen)3
Pfam Stratification Homologous
Avg pChEMBL9.37
SourceChEMBL;BindingDB
2D Structure
2D structure
Activity Profile
Target Activities (3)
Target Gene Organism Category Pfam pChEMBL Type Source
Q96KS0 EGLN2 Homo sapiens Human PF13640 9.7 IC50 ChEMBL;BindingDB
Q9GZT9 EGLN1 Homo sapiens Human PF13640 PF01753 9.7 IC50 ChEMBL;BindingDB
Q9H6Z9 EGLN3 Homo sapiens Human PF13640 8.7 IC50 ChEMBL;BindingDB