Molecule Details
InChIKeyKXZLWAAQYGMLJX-UHFFFAOYSA-N
Compound NameN-[3-(dimethylamino)propyl]-4-(5-fluoro-2,3-dihydroindol-1-yl)-5-methylpyrrolo[3,2-d]pyrimidine-6-carboxamide
Canonical SMILESCN(C)CCCNC(=O)c1cc2ncnc(N3CCc4cc(F)ccc43)c2n1C
Clinical Status Data-mined Candidate
Targets (Human+Pathogen)3
Pfam Stratification Cross-Family
Avg pChEMBL7.8
SourceChEMBL
2D Structure
2D structure
Activity Profile
Target Activities (3)
Target Gene Organism Category Pfam pChEMBL Type Source
Q9BUB5 MKNK1 Homo sapiens Human PF00069 7.9 IC50 ChEMBL
Q9HBH9 MKNK2 Homo sapiens Human PF00069 7.9 IC50 ChEMBL
P06730 EIF4E Homo sapiens Human PF01652 7.6 IC50 ChEMBL