Molecule Details
InChIKeyKXQPCNGCWDVJCL-UIOOFZCWSA-N
Canonical SMILESO=C(Nc1ccc(O[C@H]2CCNC2)c(-c2cccc(-c3nn[nH]n3)c2)c1)c1ccc(O[C@H]2CCNC2)c(-c2ccc(F)c(F)c2)c1
Clinical Status Data-mined Candidate
Targets (Human+Pathogen)2
Pfam Stratification Cross-Family
Avg pChEMBL6.08
SourceChEMBL;BindingDB
2D Structure
2D structure
Activity Profile
Target Activities (2)
Target Gene Organism Category Pfam pChEMBL Type Source
P35222 CTNNB1 Homo sapiens Human PF00514 6.2 Ki ChEMBL
O00512 BCL9 Homo sapiens Human PF11502 6.0 Ki ChEMBL;BindingDB