Molecule Details
InChIKeyKXNNHYBPDFMKQK-UHFFFAOYSA-N
Compound Name5-(2-Chloro-4-Fluorophenyl)-1-(2,6-Dichlorophenyl)-7-[1-(1-Methylethyl)piperidin-4-Yl]-3,4-Dihydroquinazolin-2(1h)-One
Canonical SMILESCC(C)N1CCC(c2cc(-c3ccc(F)cc3Cl)c3c(c2)N(c2c(Cl)cccc2Cl)C(=O)NC3)CC1
Clinical Status Data-mined Candidate
Targets (Human+Pathogen)4
Pfam Stratification Homologous
Avg pChEMBL8.86
SourceChEMBL;BindingDB
2D Structure
2D structure
Activity Profile
Target Activities (4)
Target Gene Organism Category Pfam pChEMBL Type Source
Q16539 MAPK14 Homo sapiens Human PF00069 9.2 IC50 ChEMBL;BindingDB
O15264 MAPK13 Homo sapiens Human PF00069 8.7 IC50 ChEMBL
P53778 MAPK12 Homo sapiens Human PF00069 8.7 IC50 ChEMBL
Q15759 MAPK11 Homo sapiens Human PF00069 8.7 IC50 ChEMBL