Molecule Details
InChIKeyKXMLNXWIFJZEJN-UHFFFAOYSA-N
Compound Name4-(4-cyclobutoxy-5-(2-methylbenzo[d]oxazol-6-yl)-7H-pyrrolo[2,3-d]pyrimidin-2-ylamino)-3-methoxy-N-(oxetan-3-yl)benzamide
Canonical SMILESCOc1cc(C(=O)NC2COC2)ccc1Nc1nc(OC2CCC2)c2c(-c3ccc4nc(C)oc4c3)c[nH]c2n1
Clinical Status Data-mined Candidate
Targets (Human+Pathogen)3
Pfam Stratification Homologous
Avg pChEMBL7.55
SourceChEMBL;BindingDB
2D Structure
2D structure
Activity Profile
Target Activities (3)
Target Gene Organism Category Pfam pChEMBL Type Source
P49760 CLK2 Homo sapiens Human PF00069 8.2 IC50 ChEMBL;BindingDB
P33981 TTK Homo sapiens Human PF00069 8.2 IC50 ChEMBL;BindingDB
P49759 CLK1 Homo sapiens Human PF00069 6.3 IC50 ChEMBL;BindingDB