Molecule Details
InChIKeyKXJWEXFVYFDHEI-UHFFFAOYSA-N
Compound Name2-Amino-5-(4-chloro-phenylsulfanyl)-6-methyl-3,7-dihydro-pyrrolo[2,3-d]pyrimidin-4-one
Canonical SMILESCc1[nH]c2nc(N)nc(O)c2c1Sc1ccc(Cl)cc1
Clinical Status Clinical Multi-Target
Targets (Human+Pathogen)2
Pfam Stratification Cross-Family
Avg pChEMBL6.0
SourceChEMBL;BindingDB;TTD_MultiTarget
2D Structure
2D structure
Activity Profile
Target Activities (2)
Target Gene Organism Category Pfam pChEMBL Type Source
P00374 DHFR Homo sapiens Human PF00186 6.0 pIC50 TTD_MultiTarget
P04818 TYMS Homo sapiens Human PF00303 6.0 IC50 ChEMBL;BindingDB