Molecule Details
InChIKeyKXIIKZWYFOMDJV-UHFFFAOYSA-N
Compound Name2-chloro-N-[4-(6,11-dihydropyrrolo[2,1-c][1,4]benzodiazepine-5-carbonyl)phenyl]-4-fluorobenzamide
Canonical SMILESO=C(Nc1ccc(C(=O)N2Cc3cccn3Cc3ccccc32)cc1)c1ccc(F)cc1Cl
Clinical Status Data-mined Candidate
Targets (Human+Pathogen)2
Pfam Stratification Homologous
Avg pChEMBL8.3
SourceChEMBL;BindingDB
2D Structure
2D structure
Activity Profile
Target Activities (2)
Target Gene Organism Category Pfam pChEMBL Type Source
P30518 AVPR2 Homo sapiens Human PF00001 8.4 IC50 ChEMBL;BindingDB
P37288 AVPR1A Homo sapiens Human PF00001 PF08983 8.2 IC50 ChEMBL;BindingDB