Molecule Details
InChIKeyKXICNNJQUUCJQT-UHFFFAOYSA-N
Compound Name4-[1-[3-[[2-Ethyl-5-(trifluoromethyl)pyrazole-3-carbonyl]amino]phenyl]ethylamino]quinazoline-8-carboxamide
Canonical SMILESCCn1nc(C(F)(F)F)cc1C(=O)Nc1cccc(C(C)Nc2ncnc3c(C(N)=O)cccc23)c1
Clinical Status Data-mined Candidate
Targets (Human+Pathogen)3
Pfam Stratification Homologous
Avg pChEMBL8.44
SourceChEMBL;BindingDB
2D Structure
2D structure
Activity Profile
Target Activities (3)
Target Gene Organism Category Pfam pChEMBL Type Source
Q96GD4 AURKB Homo sapiens Human PF00069 9.2 IC50 ChEMBL;BindingDB
O14965 AURKA Homo sapiens Human PF00069 8.5 IC50 ChEMBL;BindingDB
P23443 RPS6KB1 Homo sapiens Human PF00069 PF00433 7.5 IC50 ChEMBL;BindingDB