Molecule Details
InChIKeyKXDUVJWVGXIEPX-UHFFFAOYSA-N
Compound Name6-Fluoro-8-(3-fluoropiperidin-4-yl)oxy-2-([1,2,4]triazolo[4,3-a]pyridin-3-yl)quinoline
Canonical SMILESFc1cc(OC2CCNCC2F)c2nc(-c3nnc4ccccn34)ccc2c1
Clinical Status Data-mined Candidate
Targets (Human+Pathogen)2
Pfam Stratification Homologous
Avg pChEMBL7.2
SourceChEMBL;BindingDB
2D Structure
2D structure
Activity Profile
Target Activities (2)
Target Gene Organism Category Pfam pChEMBL Type Source
P11309 PIM1 Homo sapiens Human PF00069 8.1 IC50 ChEMBL;BindingDB
Q9P1W9 PIM2 Homo sapiens Human PF00069 6.3 IC50 ChEMBL;BindingDB