Molecule Details
InChIKeyKWZZDFIUKWTKDC-BULTVDLSSA-N
Compound Namemethyl N-[4-[6-chloro-5-[(1S)-1-[[(E)-3-[5-chloro-2-(tetrazol-1-yl)phenyl]prop-2-enoyl]amino]-2-phenylethyl]pyridazin-3-yl]phenyl]carbamate
Canonical SMILESCOC(=O)Nc1ccc(-c2cc([C@H](Cc3ccccc3)NC(=O)/C=C/c3cc(Cl)ccc3-n3cnnn3)c(Cl)nn2)cc1
Clinical Status Data-mined Candidate
Targets (Human+Pathogen)3
Pfam Stratification Homologous
Avg pChEMBL7.15
SourceChEMBL;BindingDB
2D Structure
2D structure
Activity Profile
Target Activities (3)
Target Gene Organism Category Pfam pChEMBL Type Source
P03951 F11 Homo sapiens Human PF00024 PF00089 8.7 Ki ChEMBL;BindingDB
P03952 KLKB1 Homo sapiens Human PF00024 PF00089 6.7 Ki ChEMBL;BindingDB
P00750 PLAT Homo sapiens Human PF00008 PF00039 PF00051 PF00089 6.0 Ki ChEMBL;BindingDB