Molecule Details
InChIKeyKWYIQYSIXKBGBV-GOSISDBHSA-N
Canonical SMILESC=CC(=O)N1CCC[C@@H](Nc2nc(Nc3ccc4c(c3)OCCOCCOCCO4)ncc2F)C1
Clinical Status Data-mined Candidate
Targets (Human+Pathogen)2
Pfam Stratification Homologous
Avg pChEMBL7.6
SourceChEMBL;BindingDB
2D Structure
2D structure
Activity Profile
Target Activities (2)
Target Gene Organism Category Pfam pChEMBL Type Source
P51813 BMX Homo sapiens Human PF00779 PF00169 PF07714 PF00017 8.1 IC50 ChEMBL;BindingDB
Q06187 BTK Homo sapiens Human PF00779 PF00169 PF07714 PF00017 PF00018 7.1 IC50 ChEMBL;BindingDB