Molecule Details
InChIKeyKWTJDPDMNWYGMB-UMSFTDKQSA-N
Canonical SMILESCCCCCN(Cc1ccc(-c2ccccc2-c2nn[nH]n2)cc1)C(=O)N1CCN(C(=O)N(c2ccccc2)c2ccccc2)[C@H](C(=O)O)C1
Clinical Status Data-mined Candidate
Targets (Human+Pathogen)2
Pfam Stratification Homologous
Avg pChEMBL7.28
SourceChEMBL;BindingDB
2D Structure
2D structure
Activity Profile
Target Activities (2)
Target Gene Organism Category Pfam pChEMBL Type Source
P30556 AGTR1 Homo sapiens Human PF00001 7.8 IC50 ChEMBL;BindingDB
P50052 AGTR2 Homo sapiens Human PF00001 6.7 IC50 ChEMBL;BindingDB