Molecule Details
InChIKeyKWLKTEPEDKFNSG-UHFFFAOYSA-N
Compound NameN-[5-(2-methoxyphenoxy)-6-[2-(propylsulfonylamino)ethoxy]-2-(3,4,5-trimethoxyphenyl)pyrimidin-4-yl]-5-propan-2-ylpyridine-2-sulfonamide
Canonical SMILESCCCS(=O)(=O)NCCOc1nc(-c2cc(OC)c(OC)c(OC)c2)nc(NS(=O)(=O)c2ccc(C(C)C)cn2)c1Oc1ccccc1OC
Clinical Status Data-mined Candidate
Targets (Human+Pathogen)2
Pfam Stratification Homologous
Avg pChEMBL7.1
SourceChEMBL;BindingDB
2D Structure
2D structure
Activity Profile
Target Activities (2)
Target Gene Organism Category Pfam pChEMBL Type Source
P24530 EDNRB Homo sapiens Human PF00001 7.6 IC50 ChEMBL;BindingDB
P25101 EDNRA Homo sapiens Human PF00001 6.6 IC50 ChEMBL;BindingDB