Molecule Details
InChIKeyKWHJKKRXFUNBAJ-QFIPXVFZSA-N
Compound Name1-amino-N-[(1S)-1-[4-(3-amino-1H-indazol-6-yl)-5-chloro-1H-imidazol-2-yl]-2-phenylethyl]isoquinoline-6-carboxamide
Canonical SMILESNc1nccc2cc(C(=O)N[C@@H](Cc3ccccc3)c3nc(-c4ccc5c(N)n[nH]c5c4)c(Cl)[nH]3)ccc12
Clinical Status Data-mined Candidate
Targets (Human+Pathogen)4
Pfam Stratification Homologous
Avg pChEMBL6.75
SourceChEMBL;BindingDB
2D Structure
2D structure
Activity Profile
Target Activities (4)
Target Gene Organism Category Pfam pChEMBL Type Source
P03951 F11 Homo sapiens Human PF00024 PF00089 7.7 Ki ChEMBL;BindingDB
P07477 PRSS1 Homo sapiens Human PF00089 6.4 Ki ChEMBL;BindingDB
P07478 PRSS2 Homo sapiens Human PF00089 6.4 Ki ChEMBL
P35030 PRSS3 Homo sapiens Human PF00089 6.4 Ki ChEMBL