Molecule Details
InChIKeyKVVMSGAISWJACO-UHFFFAOYSA-N
Compound Name1-(6-oxo-2,3,4,10b-tetrahydro-1H-pyrido[2,1-a]isoindol-10-yl)-3-pyridin-2-ylurea
Canonical SMILESO=C(Nc1ccccn1)Nc1cccc2c1C1CCCCN1C2=O
Clinical Status Data-mined Candidate
Targets (Human+Pathogen)3
Pfam Stratification Cross-Family
Avg pChEMBL7.11
SourceChEMBL;BindingDB
2D Structure
2D structure
Activity Profile
Target Activities (3)
Target Gene Organism Category Pfam pChEMBL Type Source
P06493 CDK1 Homo sapiens Human PF00069 7.1 IC50 ChEMBL;BindingDB
Q00535 CDK5 Homo sapiens Human PF00069 7.1 IC50 ChEMBL
Q15078 CDK5R1 Homo sapiens Human PF03261 7.1 IC50 ChEMBL;BindingDB