Molecule Details
InChIKeyKVVCXQIQAOOKFF-UHFFFAOYSA-N
Compound Name[4-[2-[4-[(2-Methylpyrrolo[3,4-c]quinolin-4-yl)oxymethyl]piperidin-1-yl]ethyl]phenyl]methanol
Canonical SMILESCn1cc2c(OCC3CCN(CCc4ccc(CO)cc4)CC3)nc3ccccc3c2c1
Clinical Status Data-mined Candidate
Targets (Human+Pathogen)3
Pfam Stratification Cross-Family
Avg pChEMBL7.83
SourceChEMBL;BindingDB
2D Structure
2D structure
Activity Profile
Target Activities (3)
Target Gene Organism Category Pfam pChEMBL Type Source
Q12809 KCNH2 Homo sapiens Human PF00027 PF00520 PF13426 8.0 IC50 ChEMBL;BindingDB
Q13639 HTR4 Homo sapiens Human PF00001 8.0 Ki ChEMBL;BindingDB
P28223 HTR2A Homo sapiens Human PF00001 7.5 Ki ChEMBL;BindingDB