Molecule Details
InChIKeyKVSKGMLNBAPGKH-UHFFFAOYSA-N
Compound Name3,4',5-Tribromosalicylanilide
Canonical SMILESO=C(Nc1ccc(Br)cc1)c1cc(Br)cc(Br)c1O
Clinical Status Clinical Multi-Target
Targets (Human+Pathogen)3
Pfam Stratification Cross-Family
Avg pChEMBL6.18
SourceChEMBL;TTD_MultiTarget
2D Structure
2D structure
Activity Profile
DrugBank Annotations
DrugBank ID DB20138
Drug NameTribromsalan
CAS Number87-10-5
Groups approved withdrawn
ATC Codes nan
DescriptionTribromsalan is a small molecule drug. Tribromsalan has a monoisotopic molecular weight of 446.81 Da.

Categories: Amides Amines Anilides Aniline Compounds Salicylamides
Cross-references: BindingDB: 234329 ChEBI: 127105 CHEMBL24944 Drugs Product Database (DPD): 4597 ZINC: ZINC000000538492
Target Activities (3)
Target Gene Organism Category Pfam pChEMBL Type Source
P28482 MAPK1 Homo sapiens Human PF00069 6.2 IC50 ChEMBL
Q16539 MAPK14 Homo sapiens Human PF00069 6.2 IC50 ChEMBL
P04626 ERBB2 Homo sapiens Human PF00757 PF14843 PF07714 PF01030 PF21314 Clinical TTD_MultiTarget TTD_MultiTarget