Molecule Details
InChIKeyKVJXNCXRESCVKS-UHFFFAOYSA-N
Compound Name4-(1-Ethyl-2-methylimidazol-5-yl)-2-{4-[n-(2-methoxyethyl)sulphamoyl]anilino}pyrimidine
Canonical SMILESCCn1c(-c2ccnc(Nc3ccc([S@SP3](=O)(=O)NCCOC)cc3)n2)cnc1C
Clinical Status Clinical Multi-Target
Targets (Human+Pathogen)2
Pfam Stratification Homologous
Avg pChEMBL8.4
SourceTTD_MultiTarget
2D Structure
2D structure
Activity Profile
Target Activities (2)
Target Gene Organism Category Pfam pChEMBL Type Source
P11802 CDK4 Homo sapiens Human PF00069 8.4 pIC50 TTD_MultiTarget
P24941 CDK2 Homo sapiens Human PF00069 8.4 pIC50 TTD_MultiTarget