Molecule Details
InChIKeyKVEHVMQJUPMJNA-FQEVSTJZSA-N
Compound NameN-[4-[[(1R)-4-ethynylcyclohex-3-en-1-yl]-propylamino]butyl]pyrazolo[1,5-a]pyridine-2-carboxamide
Canonical SMILESC#CC1=CC[C@H](N(CCC)CCCCNC(=O)c2cc3ccccn3n2)CC1
Clinical Status Data-mined Candidate
Targets (Human+Pathogen)3
Pfam Stratification Homologous
Avg pChEMBL7.71
SourceChEMBL;BindingDB
2D Structure
2D structure
Activity Profile
Target Activities (3)
Target Gene Organism Category Pfam pChEMBL Type Source
P35462 DRD3 Homo sapiens Human PF00001 8.5 Ki ChEMBL;BindingDB
P21917 DRD4 Homo sapiens Human PF00001 7.4 Ki ChEMBL
P14416 DRD2 Homo sapiens Human PF00001 7.2 Ki ChEMBL;BindingDB