Molecule Details
InChIKeyKUVJIFPAOJEBMN-UHFFFAOYSA-N
Compound Name7-[6-methyl-3-[(4-methyl-2-pyridinyl)methoxy]-2-pyridinyl]-2,3,4,5-tetrahydro-1H-3-benzazepine
Canonical SMILESCc1ccnc(COc2ccc(C)nc2-c2ccc3c(c2)CCNCC3)c1
Clinical Status Data-mined Candidate
Targets (Human+Pathogen)3
Pfam Stratification Cross-Family
Avg pChEMBL6.65
SourceChEMBL;BindingDB
2D Structure
2D structure
Activity Profile
Target Activities (3)
Target Gene Organism Category Pfam pChEMBL Type Source
Q96GD4 AURKB Homo sapiens Human PF00069 6.7 IC50 ChEMBL;BindingDB
Q9NQS7 INCENP Homo sapiens Human PF03941 PF12178 6.7 IC50 ChEMBL
P43405 SYK Homo sapiens Human PF07714 PF00017 6.5 IC50 ChEMBL;BindingDB