Molecule Details
InChIKeyKUQOZTZPJMJBMT-UHFFFAOYSA-N
Compound NameN-[1-[2-[4-(2-methoxyethyl)piperazin-1-yl]ethyl]pyrazol-3-yl]-2,5-dimethyl-1-phenyl-4,5-dihydropyrazolo[4,3-f]quinazolin-7-amine
Canonical SMILESCOCCN1CCN(CCn2ccc(Nc3ncc4c(n3)C(C)Cc3nn(C)c(-c5ccccc5)c3-4)n2)CC1
Clinical Status Data-mined Candidate
Targets (Human+Pathogen)3
Pfam Stratification Cross-Family
Avg pChEMBL7.79
SourceChEMBL;BindingDB
2D Structure
2D structure
Activity Profile
Target Activities (3)
Target Gene Organism Category Pfam pChEMBL Type Source
P08069 IGF1R Homo sapiens Human PF00757 PF07714 PF01030 8.5 IC50 ChEMBL;BindingDB
P06213 INSR Homo sapiens Human PF00757 PF17870 PF07714 PF01030 8.5 IC50 ChEMBL;BindingDB
O60285 NUAK1 Homo sapiens Human PF00069 6.4 IC50 ChEMBL;BindingDB