Molecule Details
InChIKeyKUJMDXMSDCLHCF-UHFFFAOYSA-N
Canonical SMILESCC(C)Oc1ccc(-c2n[nH]c3ccc(N4CCC5(CN(CC(=O)N6CC=C(c7ccc(-c8ncn(C)n8)cc7)CC6)C5)C4=O)cc23)cn1
Clinical Status Data-mined Candidate
Targets (Human+Pathogen)2
Pfam Stratification Homologous
Avg pChEMBL6.82
SourceChEMBL;BindingDB
2D Structure
2D structure
Activity Profile
Target Activities (2)
Target Gene Organism Category Pfam pChEMBL Type Source
P27361 MAPK3 Homo sapiens Human PF00069 6.8 IC50 ChEMBL;BindingDB
P28482 MAPK1 Homo sapiens Human PF00069 6.8 IC50 ChEMBL;BindingDB