Molecule Details
InChIKeyKTVJZUAZYBDWSQ-CDFUTJIBSA-N
Compound NameH-Tyr-D-Ala-Gly-Phe-Met-Ac5c-Leu-Trp-Unk
Canonical SMILESCSCC[C@H](NC(=O)[C@H](Cc1ccccc1)NC(=O)CNC(=O)[C@@H](C)NC(=O)[C@@H](N)Cc1ccc(O)cc1)C(=O)NC1(C(=O)N[C@@H](CC(C)C)C(=O)N[C@@H](Cc2c[nH]c3ccccc23)C(=O)OCc2cc(C(F)(F)F)cc(C(F)(F)F)c2)CCCC1
Clinical Status Data-mined Candidate
Targets (Human+Pathogen)2
Pfam Stratification Homologous
Avg pChEMBL9.24
SourceChEMBL;BindingDB
2D Structure
2D structure
Activity Profile
Target Activities (2)
Target Gene Organism Category Pfam pChEMBL Type Source
P25103 TACR1 Homo sapiens Human PF00001 10.2 Ki ChEMBL;BindingDB
P41143 OPRD1 Homo sapiens Human PF00001 8.3 Ki ChEMBL