Molecule Details
InChIKeyKTSCUAMGSPLOJT-VUUJKMBOSA-N
Compound Name6-(3,4-Difluoro-phenyl)-1-[(S)-5-(4-methoxycarbonyl-4-phenyl-piperidin-1-yl)-4-methyl-pentyl]-2,4-dimethyl-1,6-dihydro-pyrimidine-5-carboxylic acid methyl ester
Canonical SMILESCOC(=O)C1=C(C)N=C(C)N(CCC[C@H](C)CN2CCC(C(=O)OC)(c3ccccc3)CC2)C1c1ccc(F)c(F)c1
Clinical Status Data-mined Candidate
Targets (Human+Pathogen)3
Pfam Stratification Homologous
Avg pChEMBL7.07
SourceChEMBL;BindingDB
2D Structure
2D structure
Activity Profile
Target Activities (3)
Target Gene Organism Category Pfam pChEMBL Type Source
P35348 ADRA1A Homo sapiens Human PF00001 8.8 Ki ChEMBL;BindingDB
P35368 ADRA1B Homo sapiens Human PF00001 6.4 Ki ChEMBL;BindingDB
P25100 ADRA1D Homo sapiens Human PF00001 6.0 Ki ChEMBL;BindingDB