Molecule Details
InChIKeyKTIHAAVUVHUODX-GFCCVEGCSA-N
Compound Name(R)-4'-(3-(methylamino)pyrrolidin-1-yl)-6',7'-dihydro-5'H-spiro[cyclopentane-1,8'-quinazolin]-2'-amine
Canonical SMILESCN[C@@H]1CCN(c2nc(N)nc3c2CCCC32CCCC2)C1
Clinical Status Data-mined Candidate
Targets (Human+Pathogen)2
Pfam Stratification Homologous
Avg pChEMBL7.84
SourceChEMBL;BindingDB
2D Structure
2D structure
Activity Profile
Target Activities (2)
Target Gene Organism Category Pfam pChEMBL Type Source
Q9H3N8 HRH4 Homo sapiens Human PF00001 8.7 Ki ChEMBL;BindingDB
Q9Y5N1 HRH3 Homo sapiens Human PF00001 7.0 Ki ChEMBL;BindingDB