Molecule Details
InChIKeyKTDZCOWXCWUPEO-UHFFFAOYSA-N
Compound NameN-(2-(Cyclohexyloxy)-4-nitrophenyl)methanesulfonamide
Canonical SMILESCS(=O)(=O)Nc1ccc([N+](=O)[O-])cc1OC1CCCCC1
Clinical Status Data-mined Candidate
Targets (Human+Pathogen)2
Pfam Stratification Cross-Family
Avg pChEMBL6.49
SourceChEMBL;BindingDB
2D Structure
2D structure
Activity Profile
DrugBank Annotations
DrugBank ID DB14060
Drug NameNS-398
CAS Number123653-11-2
Groups experimental
ATC Codes nan
DescriptionNS-398 is a COX-2 inhibitor. It was developed as part of the mechanistic study of the cyclooxygenases.

Categories: Agents causing hyperkalemia Agents that produce hypertension Amides Analgesics Analgesics, Non-Narcotic Anti-Inflammatory Agents Anti-Inflammatory Agents, Non-Steroidal Antirheumatic Agents Benzene Derivatives Cyclooxygenase Inhibitors Enzyme Inhibitors Nephrotoxic agents Nitro Compounds Peripheral Nervous System Agents Sensory System Agents Sulfones Sulfur Compounds
Cross-references: BindingDB: 50029593 ChEBI: 73458 CHEMBL7162 ChemSpider: 4393 PDB: NS4 PharmGKB: PA166049196 Wikipedia: NS-398 ZINC: ZINC000003791739
Target Activities (2)
Target Gene Organism Category Pfam pChEMBL Type Source
P35354 PTGS2 Homo sapiens Human PF03098 6.8 IC50 ChEMBL;BindingDB
P11511 CYP19A1 Homo sapiens Human PF00067 6.2 IC50 ChEMBL;BindingDB
DrugBank Target Actions (3)
Target Gene Target Name Action Type
P35354 PTGS2 Prostaglandin G/H synthase 2 inhibitor enzymes
P35354 PTGS2 Prostaglandin G/H synthase 2 inhibitor targets
Q8SPQ9 PTGS2 Prostaglandin G/H synthase 2 inhibitor targets