Molecule Details
InChIKeyKSSMIJUMUAANAX-DZGCQCFKSA-N
Compound Name((1R)-6-Fluoro-8-(methylsulfonyl)-9-{(1S)-1-[4-(trifluoromethyl)phenyl]ethyl}-2,3,4,9-tetrahydro-1H-carbazol-1-yl)acetic acid
Canonical SMILESC[C@@H](c1ccc(C(F)(F)F)cc1)n1c2c(c3cc(F)cc(S(C)(=O)=O)c31)CCC[C@@H]2CC(=O)O
Clinical Status Data-mined Candidate
Targets (Human+Pathogen)3
Pfam Stratification Homologous
Avg pChEMBL7.18
SourceChEMBL;BindingDB
2D Structure
2D structure
Activity Profile
Target Activities (3)
Target Gene Organism Category Pfam pChEMBL Type Source
Q13258 PTGDR Homo sapiens Human PF00001 9.0 IC50 ChEMBL;BindingDB
P21731 TBXA2R Homo sapiens Human PF00001 6.5 Ki ChEMBL;BindingDB
P43115 PTGER3 Homo sapiens Human PF00001 6.1 Ki ChEMBL;BindingDB