Molecule Details
InChIKeyKSIKWQAAQUDISH-UHFFFAOYSA-N
Compound Name5-{[(4-Amino-3-chloro-5-iodophenyl)sulfonyl]amino}-1,3,4-thiadiazole-2-sulfonamide
Canonical SMILESNc1c(Cl)cc(S(=O)(=O)Nc2nnc(S(N)(=O)=O)s2)cc1I
Clinical Status Clinical Multi-Target
Targets (Human+Pathogen)3
Pfam Stratification Cross-Family
Avg pChEMBL9.0
SourceChEMBL;BindingDB;TTD_MultiTarget
2D Structure
2D structure
Activity Profile
Target Activities (3)
Target Gene Organism Category Pfam pChEMBL Type Source
P00918 CA2 Homo sapiens Human PF00194 9.1 Ki ChEMBL;BindingDB
P18505 GABRB1 Homo sapiens Human PF02931 PF02932 9.1 pIC50 TTD_MultiTarget
P00915 CA1 Homo sapiens Human PF00194 8.8 Ki ChEMBL;BindingDB