Molecule Details
InChIKeyKSDORXSBAJOQKH-UHFFFAOYSA-N
Compound Name2-(1h-Indazol-5-yl)-3-phenylimidazo[1,2-a]pyrimidine
Canonical SMILESc1ccc(-c2c(-c3ccc4[nH]ncc4c3)nc3ncccn23)cc1
Clinical Status Data-mined Candidate
Targets (Human+Pathogen)3
Pfam Stratification Homologous
Avg pChEMBL7.56
SourceChEMBL;BindingDB
2D Structure
2D structure
Activity Profile
Target Activities (3)
Target Gene Organism Category Pfam pChEMBL Type Source
O75116 ROCK2 Homo sapiens Human PF25346 PF00069 PF08912 8.2 Ki ChEMBL;BindingDB
P49841 GSK3B Homo sapiens Human PF00069 8.0 Ki ChEMBL;BindingDB
P11309 PIM1 Homo sapiens Human PF00069 6.5 Ki ChEMBL;BindingDB