Molecule Details
InChIKeyKRWCFCQJKXIENS-UHFFFAOYSA-N
Compound Name5-(2-amino-4-pyridinyl)-2-methyl-N-(thiophen-3-ylmethyl)-7H-pyrrolo[2,3-d]pyrimidin-4-amine
Canonical SMILESCc1nc(NCc2ccsc2)c2c(-c3ccnc(N)c3)c[nH]c2n1
Clinical Status Data-mined Candidate
Targets (Human+Pathogen)3
Pfam Stratification Homologous
Avg pChEMBL8.24
SourceChEMBL;BindingDB
2D Structure
2D structure
Activity Profile
Target Activities (3)
Target Gene Organism Category Pfam pChEMBL Type Source
Q9Y463 DYRK1B Homo sapiens Human PF00069 9.0 IC50 ChEMBL;BindingDB
Q13627 DYRK1A Homo sapiens Human PF00069 7.9 IC50 ChEMBL;BindingDB
Q92630 DYRK2 Homo sapiens Human PF00069 7.8 IC50 ChEMBL;BindingDB