Molecule Details
InChIKeyKRVYWSXTKLCPHD-IRXDYDNUSA-N
Compound Name(6S,7S)-6-[4-(3,5-difluorophenyl)-3,6-dihydro-2H-pyridine-1-carbonyl]-N-hydroxy-5-azaspiro[2.5]octane-7-carboxamide
Canonical SMILESO=C(NO)[C@H]1CC2(CC2)CN[C@@H]1C(=O)N1CC=C(c2cc(F)cc(F)c2)CC1
Clinical Status Clinical Multi-Target
Targets (Human+Pathogen)3
Pfam Stratification Cross-Family
Avg pChEMBL7.2
SourceChEMBL;BindingDB;TTD_MultiTarget
2D Structure
2D structure
Activity Profile
Target Activities (3)
Target Gene Organism Category Pfam pChEMBL Type Source
P08253 MMP2 Homo sapiens Human PF00040 PF00045 PF00413 7.8 pIC50 TTD_MultiTarget
O14672 ADAM10 Homo sapiens Human PF21299 PF00200 PF13574 7.7 IC50 ChEMBL;BindingDB
P14780 MMP9 Homo sapiens Human PF00040 PF00045 PF00413 6.0 IC50 ChEMBL;BindingDB