Molecule Details
InChIKeyKRVOJOCLBAAKSJ-UHFFFAOYSA-N
Compound NameN-(1-benzyl-2-methylpyrrolidin-3-yl)-5-chloro-2-methoxy-4-(methylamino)benzamide
Canonical SMILESCNc1cc(OC)c(C(=O)NC2CCN(Cc3ccccc3)C2C)cc1Cl
Clinical Status Data-mined Candidate
Targets (Human+Pathogen)4
Pfam Stratification Cross-Family
Avg pChEMBL8.74
SourceChEMBL;BindingDB
2D Structure
2D structure
Activity Profile
Target Activities (4)
Target Gene Organism Category Pfam pChEMBL Type Source
P21917 DRD4 Homo sapiens Human PF00001 9.0 Ki ChEMBL;BindingDB
P35462 DRD3 Homo sapiens Human PF00001 9.0 Ki ChEMBL
P14416 DRD2 Homo sapiens Human PF00001 8.8 Ki ChEMBL
Q5BJF2 TMEM97 Homo sapiens Human PF05241 8.1 Ki ChEMBL