Molecule Details
InChIKeyKRTIYQIPSAGSBP-KLAILNCOSA-N
Compound Name(2R)-N-(4-Chlorophenyl)-2-(cis-4-(6-fluoro-4-quinolinyl)cyclohexyl)propanamide
Canonical SMILESC[C@@H](C(=O)Nc1ccc(Cl)cc1)C1CCC(c2ccnc3ccc(F)cc23)CC1
Clinical Status Data-mined Candidate
Targets (Human+Pathogen)2
Pfam Stratification Cross-Family
Avg pChEMBL7.44
SourceBindingDB;ChEMBL
2D Structure
2D structure
Activity Profile
Target Activities (2)
Target Gene Organism Category Pfam pChEMBL Type Source
P14902 IDO1 Homo sapiens Human PF01231 8.7 IC50 ChEMBL;BindingDB
P11712 CYP2C9 Homo sapiens Human PF00067 6.1 IC50 BindingDB