Molecule Details
InChIKeyKPUBBCGAMBGWSV-UHFFFAOYSA-N
Compound NamePyrazolo[4,3-h]quinazoline-3-carboxamide, 21
Canonical SMILESCn1nc(C(=O)NCc2ccccc2)c2c1-c1nc(Nc3ccccc3)ncc1CC2
Clinical Status Clinical Multi-Target
Targets (Human+Pathogen)2
Pfam Stratification Homologous
Avg pChEMBL6.43
SourceChEMBL;BindingDB;TTD_MultiTarget
2D Structure
2D structure
Activity Profile
Target Activities (2)
Target Gene Organism Category Pfam pChEMBL Type Source
O14965 AURKA Homo sapiens Human PF00069 6.4 IC50 ChEMBL;BindingDB
P24941 CDK2 Homo sapiens Human PF00069 6.4 pIC50 TTD_MultiTarget