Molecule Details
InChIKeyKPRXKFKHZVTBIT-UHFFFAOYSA-N
Compound Name6-Methyl-29-oxo-19-oxa-2,6,10,12-tetrazahexacyclo[18.5.2.12,5.114,18.08,12.023,26]nonacosa-8,10,14(28),15,17,20(27),21,23(26)-octaene-17-carbonitrile
Canonical SMILESCN1Cc2cncn2Cc2ccc(C#N)c(c2)Oc2ccc3c(c2)C(CC3)N2CCC1C2=O
Clinical Status Clinical Multi-Target
Targets (Human+Pathogen)2
Pfam Stratification Cross-Family
Avg pChEMBL8.85
SourceChEMBL;TTD_MultiTarget
2D Structure
2D structure
Activity Profile
Target Activities (2)
Target Gene Organism Category Pfam pChEMBL Type Source
P49354 FNTA Homo sapiens Human PF01239 8.8 pIC50 TTD_MultiTarget
P49356 FNTB Homo sapiens Human PF00432 8.8 IC50 ChEMBL