Molecule Details
InChIKeyKPJVSWMSLFZHBU-NLHRSOKXSA-N
Compound NameAc-Leu-Asn-Glu-His-Val-Arg-Asp-Gln-Tyr-Pro-Gly-Leu-Asp-Glu-Met-Trp-Lys-Arg-Asp-Phe-Pro-Arg-Glu-Ser-Ile-Arg-Thr-His-Thr-Ala-NH2
Canonical SMILESCC[C@H](C)[C@H](NC(=O)[C@H](CO)NC(=O)[C@H](CCC(=O)O)NC(=O)[C@H](CCCNC(=N)N)NC(=O)[C@@H]1CCCN1C(=O)[C@H](Cc1ccccc1)NC(=O)[C@H](CC(=O)O)NC(=O)[C@H](CCCNC(=N)N)NC(=O)[C@H](CCCCN)NC(=O)[C@H](Cc1c[nH]c2ccccc12)NC(=O)[C@H](CCSC)NC(=O)[C@H](CCC(=O)O)NC(=O)[C@H](CC(=O)O)NC(=O)[C@H](CC(C)C)NC(=O)CNC(=O)[C@@H]1CCCN1C(=O)[C@H](Cc1ccc(O)cc1)NC(=O)[C@H](CCC(N)=O)NC(=O)[C@H](CC(=O)O)NC(=O)[C@H](CCCNC(=N)N)NC(=O)[C@@H](NC(=O)[C@H](Cc1cnc[nH]1)NC(=O)[C@H](CCC(=O)O)NC(=O)[C@H](CC(N)=O)NC(=O)[C@H](CC(C)C)NC(C)=O)C(C)C)C(=O)N[C@@H](CCCNC(=N)N)C(=O)N[C@H](C(=O)N[C@@H](Cc1cnc[nH]1)C(=O)N[C@H](C(=O)N[C@@H](C)C(N)=O)[C@@H](C)O)[C@@H](C)O
Clinical Status Data-mined Candidate
Targets (Human+Pathogen)3
Pfam Stratification Cross-Family
Avg pChEMBL6.53
SourceChEMBL
2D Structure
2D structure
Activity Profile
Target Activities (3)
Target Gene Organism Category Pfam pChEMBL Type Source
P21730 C5AR1 Homo sapiens Human PF00001 6.9 Kd ChEMBL
Q9P296 C5AR2 Homo sapiens Human PF00001 6.6 Kd ChEMBL
P01031 C5 Homo sapiens Human PF00207 PF07703 PF07677 PF01821 PF21309 PF17790 PF01835 PF17791 PF17789 PF01759 PF07678 6.1 Kd ChEMBL