Molecule Details
InChIKeyKPDOBADQSPMGFP-OELJMHDBSA-O
Compound Name[(1R)-1-[(10S,13S,16S)-16-[[(2S)-2-[[(2S)-1-acetylpyrrolidine-2-carbonyl]amino]-4-methylpentanoyl]amino]-13-(hydroxymethyl)-9,12,15-trioxo-19-(8-phenyloctyl)-8,11,14,19-tetraza-1-azoniabicyclo[16.2.1]henicosa-1(20),18(21)-dien-10-yl]ethyl] dihydrogen phosphate
Canonical SMILESCC(=O)N1CCC[C@H]1C(=O)N[C@@H](CC(C)C)C(=O)N[C@H]1Cc2c[n+](cn2CCCCCCCCc2ccccc2)CCCCCCNC(=O)[C@H]([C@@H](C)OP(=O)(O)O)NC(=O)[C@H](CO)NC1=O
Clinical Status Data-mined Candidate
Targets (Human+Pathogen)3
Pfam Stratification Homologous
Avg pChEMBL7.3
SourceChEMBL;BindingDB
2D Structure
2D structure
Activity Profile
Target Activities (3)
Target Gene Organism Category Pfam pChEMBL Type Source
P53350 PLK1 Homo sapiens Human PF00069 PF00659 7.8 IC50 ChEMBL;BindingDB
Q9H4B4 PLK3 Homo sapiens Human PF00069 PF00659 7.1 IC50 ChEMBL;BindingDB
Q9NYY3 PLK2 Homo sapiens Human PF00069 PF00659 7.0 IC50 ChEMBL;BindingDB