Molecule Details
InChIKeyKOARITDFMAWYET-UHFFFAOYSA-N
Compound Name4-[3-(4-piperazin-1-ylphenyl)-1H-indol-6-yl]phenol
Canonical SMILESOc1ccc(-c2ccc3c(-c4ccc(N5CCNCC5)cc4)c[nH]c3c2)cc1
Clinical Status Data-mined Candidate
Targets (Human+Pathogen)3
Pfam Stratification Homologous
Avg pChEMBL7.81
SourceChEMBL;BindingDB
2D Structure
2D structure
Activity Profile
Target Activities (3)
Target Gene Organism Category Pfam pChEMBL Type Source
P11309 PIM1 Homo sapiens Human PF00069 8.4 IC50 ChEMBL;BindingDB
Q86V86 PIM3 Homo sapiens Human PF00069 7.7 IC50 ChEMBL;BindingDB
Q9P1W9 PIM2 Homo sapiens Human PF00069 7.4 IC50 ChEMBL;BindingDB