Molecule Details
InChIKeyKNQRBVIESPJOCL-TZIWHRDSSA-N
Canonical SMILESCOc1ccc(CNc2nc3c(OC)cc(F)cc3c3nc([C@@H]4C[C@@H](F)CN(c5cnn(CC(C)(C)O)c5)C4)nn23)c(OC)c1
Clinical Status Data-mined Candidate
Targets (Human+Pathogen)2
Pfam Stratification Homologous
Avg pChEMBL7.94
SourceChEMBL;BindingDB
2D Structure
2D structure
Activity Profile
Target Activities (2)
Target Gene Organism Category Pfam pChEMBL Type Source
P29274 ADORA2A Homo sapiens Human PF00001 9.1 IC50 ChEMBL;BindingDB
P29275 ADORA2B Homo sapiens Human PF00001 6.8 IC50 ChEMBL;BindingDB