Molecule Details
InChIKeyKNOAXFIYIPQVPI-UHFFFAOYSA-N
Compound Name(1R,2R and 1S,2S)-N-(3-Methyl-1,2-thiazol-5-yl)-2-[4-(1H-pyrazol-5-yl)benzoyl]cyclohexanecarboxamide
Canonical SMILESCc1cc(NC(=O)C2CCCCC2C(=O)c2ccc(-c3ccn[nH]3)cc2)sn1
Clinical Status Data-mined Candidate
Targets (Human+Pathogen)3
Pfam Stratification Cross-Family
Avg pChEMBL7.64
SourceChEMBL;BindingDB
2D Structure
2D structure
Activity Profile
Target Activities (3)
Target Gene Organism Category Pfam pChEMBL Type Source
P09917 ALOX5 Homo sapiens Human PF00305 PF01477 7.6 IC50 ChEMBL;BindingDB
P20292 ALOX5AP Homo sapiens Human PF01124 7.6 IC50 ChEMBL
P39748 FEN1 Homo sapiens Human PF00867 PF00752 7.6 IC50 ChEMBL