Molecule Details
InChIKeyKNAZBXXUUKXFRJ-UHFFFAOYSA-N
Canonical SMILESCOC(=O)N1CC2(CN(Cc3ccc(-c4cccc(-c5cccc(-c6ccc(CN7CC8(C7)CN(C(=O)OC)C8)c(OC)n6)c5Cl)c4Cl)nc3OC)C2)C1
Clinical Status Data-mined Candidate
Targets (Human+Pathogen)2
Pfam Stratification Cross-Family
Avg pChEMBL6.22
SourceChEMBL;BindingDB
2D Structure
2D structure
Activity Profile
Target Activities (2)
Target Gene Organism Category Pfam pChEMBL Type Source
Q9BQ51 PDCD1LG2 Homo sapiens Human PF22705 6.2 IC50 ChEMBL;BindingDB
Q9NZQ7 CD274 Homo sapiens Human PF08205 PF07686 6.2 IC50 ChEMBL