Molecule Details
InChIKeyKMYJUKQUMDPSJU-UHFFFAOYSA-N
Compound Name8-[(3,4-dichlorophenyl)methyl]-1,3-dimethyl-7,9-dihydro-6H-purino[7,8-a]pyrazine-2,4-dione
Canonical SMILESCn1c(=O)c2c(nc3n2CCN(Cc2ccc(Cl)c(Cl)c2)C3)n(C)c1=O
Clinical Status Data-mined Candidate
Targets (Human+Pathogen)2
Pfam Stratification Cross-Family
Avg pChEMBL6.4
SourceChEMBL;BindingDB
2D Structure
2D structure
Activity Profile
Target Activities (2)
Target Gene Organism Category Pfam pChEMBL Type Source
P27338 MAOB Homo sapiens Human PF01593 6.7 IC50 ChEMBL;BindingDB
P30542 ADORA1 Homo sapiens Human PF00001 6.1 Ki ChEMBL;BindingDB