Molecule Details
InChIKeyKMRKVWIQPVPEED-UHFFFAOYSA-N
Compound Name4-[[[5-[5-(6-chloro-1H-benzimidazol-2-yl)-2-pyridinyl]-2-pyridinyl]amino]methyl]benzoic acid
Canonical SMILESO=C(O)c1ccc(CNc2ccc(-c3ccc(-c4nc5cc(Cl)ccc5[nH]4)cn3)cn2)cc1
Clinical Status Data-mined Candidate
Targets (Human+Pathogen)2
Pfam Stratification Cross-Family
Avg pChEMBL8.31
SourceChEMBL;BindingDB
2D Structure
2D structure
Activity Profile
Target Activities (2)
Target Gene Organism Category Pfam pChEMBL Type Source
P10632 CYP2C8 Homo sapiens Human PF00067 8.6 IC50 ChEMBL;BindingDB
O75907 DGAT1 Homo sapiens Human PF03062 8.0 IC50 ChEMBL;BindingDB